LIttoral ENvironnement et Sociétés (LIENSs) - UMR 7266

Thiéry Valérie

Équipe de rattachement : BCBS
Statut : Chercheur
valerie.thiery*at*univ-lr.fr
Tél. : +33 (O)5 46 45 82 76

Enseignant-chercheur, Professeur
Université de La Rochelle
Section de Recherche : CNU 32
Institut scientifique du CNRS référent : INEE

Mots clés : Hétérocycles, alcaloïde, chimie verte, micro-onde

Responsable du groupe de chimie organique
Correspondant Hygiène et Sécurité de LIENSs-CURIE

Thèmes de Recherche.

Chimie hétérocyclique (N,O,S), étude de la réactivité des iminodithiazoles

Synthèse d’analogues d’alcaloïdes marins à visée antitumorales

Synthèse d’inhibiteurs de kinases

Chimie assistée- par micro-ondes : nouvelles méthodologies de synthèse, extraction

Synthèse asymétrique

Liste des publications :

56 résultats

2022

Article dans une revue

From benzofuro-, benzothieno- and 10-methylindolo-[2,3-b]-fused benzothiopyrano[4,3,2-de]quinolines to the corresponding benzothiopyrano[4,3,2-de]1,8-naphthyridines: synthesis and properties of these hexacyclic heteroaromatic compounds

Nicolas Mast , William Erb , Lionel Nauton , Pascale Moreau , Olivier Mongin , Thierry Roisnel , Margaux Macaigne , Thomas Robert , Stéphane Bach , Laurent Picot , Valérie Thiéry , Jean-Pierre Hurvois , Florence Mongin

New Journal of Chemistry, 2022, 47 (1), pp.258-283. ⟨10.1039/D2NJ04567B⟩

Bisphosphonylallenes as Suitable Scaffolds for Unprecedented 4,5-Diphosphonyldihydropyridazines and 3,4-Diphosphonylpyrroles Displaying Antimelanoma Activity

Kmar Abaid , William Erb , David Virieux , Laurent Picot , Benjamin Musnier , Valérie Thiéry , Thierry Roisnel , Florence Mongin , Soufiane Touil

ACS Omega, 2022, 7 (43), pp.38894-38901. ⟨10.1021/acsomega.2c04619⟩

Archaea Carotenoids: Natural Pigments with Unexplored Innovative Potential

Antoine Grivard , Isabelle Goubet , Luiz Miranda de Souza Duarte Filho , Valérie Thiéry , Sylvie Chevalier , Raimundo Gonçalves de Oliveira-Junior , Noureddine El Aouad , Jackson Roberto Guedes da Silva Almeida , Przemysław Sitarek , Lucindo José Quintans-Junior , Raphaël Grougnet , Hélène Agogué , Laurent Picot

Marine drugs, 2022, 20 (8), pp.524. ⟨10.3390/md20080524⟩

Archaea Carotenoids: Natural Pigments with Unexplored Innovative Potential

Antoine Grivard , Isabelle Goubet , Luiz Miranda de Souza Duarte Filho , Valérie Thiéry , Sylvie Chevalier , Raimundo Gonçalves de Oliveira-Junior , Noureddine El Aouad , Jackson Roberto Guedes da Silva Almeida , Przemysław Sitarek , Lucindo José Quintans-Junior , Raphaël Grougnet , Hélène Agogué , Laurent Picot

Marine drugs, 2022, 20 (8), pp.524. ⟨10.3390/md20080524⟩

Alterins, a new family of marine antibacterial cyclolipopeptides

Clément Offret , Héléna Cuny , Pierre-Edouard Bodet , Florie Desriac , Camille Jegou , Alexis Bazire , Romain Chevrot , Valérie Thiery , Benjamin Brillet , Yannick Fleury

International Journal of Antimicrobial Agents, 2022, pp.106514. ⟨10.1016/j.ijantimicag.2021.106514⟩

2021

Article dans une revue

Thiazolo[5,4- f ]quinoxalines, Oxazolo[5,4- f ]quinoxalines and Pyrazino[ b,e ]isatins: Synthesis from 6-Aminoquinoxalines and Properties

Frédéric Lassagne , Joshua M. Sims , William Erb , Olivier Mongin , Nicolas Richy , Nour El Osmani , Ziad Fajloun , Laurent Picot , Valérie Thiéry , Thomas Robert , Stéphane Bach , Vincent Dorcet , Thierry Roisnel , Florence Mongin

European Journal of Organic Chemistry, 2021, 2021 (19), pp.2756-2763. ⟨10.1002/ejoc.202100362⟩

The Franco-Brazilian network on natural products (FB2NP): a new network promoting cooperation and exchanges in natural products research

Jackson Almeida , Raphaël Grougnet , Lucindo Quintans , Marc Feuilloley , Thomas Robert , Stéphane Bach , Raimundo Oliveira , Valérie Thiéry , Jean-Pierre Bazureau , Florence Mongin , Marina Kritsanida , Vincent Sol , Vicente Costa , Nathalie Bourgougnon , Pascal Marchand , Laurent Picot , Sylvie Chevalier

Química Nova, 2021, ⟨10.21577/0100-4042.20170847⟩

Iodothiophenes and Related Compounds as Coupling Partners in Copper-Mediated N-Arylation of Anilines

Salima Bouarfa , Ghenia Bentabed-Ababsa , William Erb , Laurent Picot , Valérie Thiéry , Thierry Roisnel , Vincent Dorcet , Florence Mongin

Synthesis: Journal of Synthetic Organic Chemistry, 2021, 53 (07), pp.1271-1284. ⟨10.1055/s-0040-1706542⟩

THE FRANCO-BRAZILIAN NETWORK ON NATURAL PRODUCTS (FB2NP): A NEW NETWORK PROMOTING COOPERATION AND EXCHANGES IN NATURAL PRODUCTS RESEARCH

Jackson Almeida , Raphaël Grougnet , Lucindo Quintans , Sylvie Chevalier , Marc Feuilloley , Thomas Robert , Stéphane Bach , Raimundo Oliveira , Valérie Thiéry , Jean-Pierre Bazureau , Florence Mongin , Marina Kritsanida , Vincent Sol , Vicente Costa , Nathalie Bourgougnon , Pascal Marchand , Laurent Picot

Química Nova, 2021, ⟨10.21577/0100-4042.20170847⟩

2020

Article dans une revue

2-Aminobenzaldehyde, a common precursor to acridines and acridones endowed with bioactivities

Sarah Zeghada , Ghenia Bentabed-Ababsa , Olivier Mongin , William Erb , Laurent Picot , Valérie Thiéry , Thierry Roisnel , Vincent Dorcet , Florence Mongin

Tetrahedron, 2020, 76 (38), pp.131435. ⟨10.1016/j.tet.2020.131435⟩

Carotenoids from Rhodomonas salina Induce Apoptosis and Sensitize A2058 Melanoma Cells to Chemotherapy

Raimundo Gonçalves de Oliveira-Júnior , Elodie Nicolau , Antoine Bonnet , Grégoire Prunier , Laureen Beaugeard , Nicolas Joguet , Valérie Thiéry , Laurent Picot

Revista Brasileira de Farmacognosia, 2020, 30 (2), pp.155-168. ⟨10.1007/s43450-020-00036-2⟩

Functionalization of 9-thioxanthone at the 1-position: From arylamino derivatives to [1]benzo(thio)pyrano[4,3,2-de]benzothieno[2,3-b]quinolines of biological interest

Nahida Mokhtari Brikci-Nigassa , Lionel Nauton , Pascale Moreau , Olivier Mongin , Raphael E Duval , Laurent Picot , Valérie Thiery , Mohamed Souab , Blandine Baratte , Sandrine Ruchaud , Stéphane Bach , Rémy Le Guével , Ghenia Bentabed-Ababsa , William Erb , Thierry Roisnel , Vincent Dorcet , Florence Mongin

Bioorganic Chemistry, 2020, 94, pp.103347. ⟨10.1016/j.bioorg.2019.103347⟩

2019

Article dans une revue

Characterisation of the anti-migratory activity of the 6-bromoindirubin-3’oxime (BIO) derivative VTIND42 in patient-derived GBM subpopulations

Samuel Peat , Anke Bruning-Richardson , Laurent Meijer , Sean Lawler , Valérie Thiéry , Ruth Morton

Neuro-Oncology, 2019, 21 (Supplement_4), pp.iv6-iv7. ⟨10.1093/neuonc/noz167.026⟩

Crystal Structure of 6,7-Dihydro-5a,7a,13,14-tetraaza-pentaphene-5,8-dione

Jean Guillon , Maria de Fatima Pereira-Rosenfeld , Noël Pinaud , Thierry Besson , Valérie Thiéry , Laurent Picot , Mathieu Marchivie

X-Ray Structure Analysis Online, 2019, 35 (10), pp.57-59. ⟨10.2116/xraystruct.35.57⟩

2018

Article dans une revue

Complete Genome Sequence of the Polymyxin E (Colistin)-Producing Paenibacillus sp. Strain B-LR

Caroline Salsano , Sandrine Didelot , Fatoumata Tambadou , Thibault Caradec , Valérie Sopena , Cyrille Barthélémy , Valérie Thiéry , Romain Chevrot

Microbiology Resource Announcements, 2018, 7 (23), ⟨10.1128/MRA.01013-18⟩

From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines

Frédéric Lassagne , Timothy Langlais , Elsa Caytan , Emmanuelle Limanton , Ludovic Paquin , Manon Boullard , Coline Courtel , Idriss Curbet , Clément Gédéon , Julien Lebreton , Laurent Picot , Valérie Thiéry , Mohamed Souab , Blandine Baratte , Sandrine Ruchaud , Stéphane Bach , Thierry Roisnel , Florence Mongin

Molecules, 2018, 23 (11), pp.2961. ⟨10.3390/molecules23112961⟩

Sensitization of tumor cells to chemotherapy by natural products: a systematic review of preclinical data and molecular mechanisms

Raimundo Gonçalves de Oliveira Júnior , Christiane Adrielly Alves Ferraz , Jackson Roberto Guedes da Silva Almeida , Raphäel Grougnet , Valérie Thiéry , Laurent Picot

Fitoterapia, 2018, 129, pp.383-400. ⟨10.1016/j.fitote.2018.02.025⟩

Synthesis of 2-Mercapto-(2-Oxoindolin-3-Ylidene)Acetonitriles from 3-(4-Chloro-5H-1,2,3-Dithiazol-5-Ylidene)Indolin-2-ones

Boris Letribot , Régis Delatouche , Hervé Rouillard , Antoine Bonnet , Jean-René Chérouvrier , Lisianne Domon , Thierry Besson , Valérie Thiéry

Molecules, 2018, 23 (6), pp.1390. ⟨10.3390/molecules23061390⟩

2-Aminophenones, a common precursor to N-aryl isatins and acridines endowed with bioactivities

Nahida Mokhtari Brikci-Nigassa , Ghenia Bentabed-Ababsa , William Erb , Floris Chevallier , Laurent Picot , Lucille Vitek , Audrey Fleury , Valérie Thiéry , Mohamed Souab , Thomas Robert , Sandrine Ruchaud , Stéphane Bach , Thierry Roisnel , Florence Mongin

Tetrahedron, 2018, 74 (15), pp.1785-1801. ⟨10.1016/j.tet.2018.02.038⟩

Zeaxanthin from Porphyridium purpureum induces apoptosis in human melanoma cells expressing the oncogenic BRAF V600E mutation and sensitizes them to the BRAF inhibitor vemurafenib

Camille Juin , Raimundo Gonçalves de Oliveira Junior , Audrey Fleury , Chloé Oudinet , Lior Pytowski , Jean-Baptiste Bérard , Elodie Nicolau , Valérie Thiéry , Isabelle Lanneluc , Laureen Beaugeard , Grégoire Prunier , Jackson Roberto Guedes da Silva Almeida , Laurent Picot

Revista Brasileira de Farmacognosia, 2018, 28 (4), pp.457-467. ⟨10.1016/j.bjp.2018.05.009⟩

2017

Article dans une revue

Synthesis of novel heterocyclic fused pyrimidin-4-one derivatives from imino-1,2,3-dithiazoles

Maria de Fatima Pereira , Elena Sarghe , Hervé Rouillard , Lisianne Domon , Jean-René Chérouvrier , Valérie Thiéry , Jacques Royer

ARKIVOC - Online Journal of Organic Chemistry, 2017, 2017 (3), pp.335-345. ⟨10.24820/ark.5550190.p010.256⟩

Antimelanoma activity of Heterocapsa triquetra pigments

Quentin Haguet , Antoine Bonnet , Jean-Baptiste Bérard , Joelle Goldberg , Nicolas Joguet , Audrey Fleury , Valérie Thiéry , Laurent Picot

Algal Research - Biomass, Biofuels and Bioproducts, 2017, 25, pp.207 - 215. ⟨10.1016/j.algal.2017.04.034⟩

2016

Article dans une revue

Improved racemate resolution of pentan-2-ol and trans-(Z)-cyclooct-5-ene-1,2-diol by lipase catalysis

Marianne Graber , Hervé Rouillard , Régis Delatouche , Najla Fniter , Belsem Belkhiria , Antoine Bonnet , Lisiane Domon , Valérie Thiéry

Journal of Biotechnology, 2016, 238, pp.60-68. ⟨10.1016/j.jbiotec.2016.09.010⟩

Could Fucoxanthin Interaction with Lipid Rafts Mediate its Cytotoxicity in Cancer Cells?

Raimundo Gonçalves Oliveira-Junior , Valérie Thiéry , Odile Sergent , Martine Chevanne , Laurent Picot

Journal of Oceanography and Marine Research, 2016, 4 (1), pp.1000144. ⟨10.4172/jomr.1000144⟩

2015

Article dans une revue

Azine and Diazine Functionalization Using 2,2,6,6-Tetramethylpiperidino-Based Lithium–Metal Combinations: Application to the Synthesis of 5,9-Disubstituted Pyrido[3′,2′:4,5]pyrrolo[1,2-c] pyrimidines

Nada Marquise , Tan Tai Nguyen , Floris Chevallier , Laurent Picot , Valérie Thiéry , Olivier Lozach , Stéphane Bach , Sandrine Ruchaud , Florence Mongin

SYNLETT, 2015, 26 (20), pp.2811-2816. ⟨10.1055/s-0035-1560496⟩

Deproto-metallation of N-arylated pyrroles and indoles using a mixed lithium–zinc base and regioselectivity-computed CH acidity relationship

Mohamed Yacine Ameur Messaoud , Ghenia Bentabed-Ababsa , Madani Hedidi , Aïcha Derdour , Floris Chevallier , Yury S. Halauko , Oleg A. Ivashkevich , Vadim E. Matulis , Laurent Picot , Valérie Thiéry , Thierry Roisnel , Vincent Dorcet , Florence Mongin

Beilstein Journal of Organic Chemistry, 2015, 11, pp.1475-1485. ⟨10.3762/bjoc.11.160⟩

Caractérisations analytiques des extraits colorants des plantes tinctoriales d'Afrique Centrale

A.B. Madiélé , Jean-Michel Zhao , Valérie Thiéry , Huguette Agnaniet , Christine Brunet , Marianne Graber , J. M. Ouamba

Lebanese Science Journal, 2015, 16, pp.33-44

Characterization of the colistin (polymyxin E1 and E2) biosynthetic gene cluster.

Fatoumata Tambadou , Thibault Caradec , Anne-Laure Gagez , Antoine Bonnet , Valérie Sopena , Nicolas Bridiau , Valérie Thiéry , Sandrine Didelot, , Cyrille Barthélémy , Romain Chevrot

Archives of Microbiology, 2015, 197 (4), pp.521-532. ⟨10.1007/s00203-015-1084-5⟩

Microwave-Assisted Extraction of Phycobiliproteins from Porphyridium purpureum.

Camille Juin , Jean-René Chérouvrier , Valérie Thiery , Anne-Laure Gagez , Jean-Baptiste Bérard , Nicolas, Joguet , Raymond Kaas , Jean-Paul Cadoret , Laurent Picot

Biotechnology and Applied Biochemistry, 2015, ⟨10.1007/s12010-014-1250-2⟩

UPLC-MSE Profiling of Phytoplankton Metabolites: Application to the Identification of Pigments and Structural Analysis of Metabolites in Porphyridium purpureum

Camille Juin , Antoine Bonnet , Elodie Nicolau , Jean-Baptiste Bérard , Devillers, Romain , Valérie Thiéry , Jean-Paul Cadoret , Laurent Picot

Marine drugs, 2015, 13 (4), pp.1541-2558. ⟨10.3390/md13042541⟩

2014

Article dans une revue

Microwave-Assisted Kinetic Resolution of Homochiral (Z)-Cyclooct-5-ene-1,2-diol and (Z)-2-Acetoxycyclooct-4-enyl Acetate Using Lipases

Hervé Rouillard , Emmanuel Deau , Lisiane Domon , Jean-René Chérouvrier , Marianne Graber , Valérie Thiéry

Molecules, 2014, 19, pp.9215-9227. ⟨10.3390/molecules19079215⟩

Novel nonribosomal peptide synthetase (NRPS) genes sequenced from intertidal mudflat bacteria

Fatoumata Tambadou , Isabelle Lanneluc , Sophie Sablé , Géraldine Klein , Ibtissem Doghri , Valérie Sopena , Sandrine Didelot , Cyrille Barthélémy , Valérie Thiéry , Romain Chevrot

FEMS Microbiology Letters, 2014, pp.n/a-n/a. ⟨10.1111/1574-6968.12532⟩

Synthesis of C,N'-linked bis-heterocycles using a deprotometalation-iodination-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells

Madani Hedidi , Ghenia Bentabed-Ababsa , Aicha Derdour , Thierry Roisnel , Vincent Dorcet , Floris Chevallier , Laurent Picot , Valérie Thiery , Mongin Florence

Bioorganic and Medicinal Chemistry, 2014, 22 (13), pp.3498-3507. ⟨10.1016/j.bmc.2014.04.028⟩

2013

Article dans une revue

Synthesis of azafluorenones and related compounds using deprotocupration-aroylation followed by intramolecular direct arylation

Nada Marquise , Philip J. Harford , Floris Chevallier , Thierry Roisnel , Vincent Dorcet , Anne-Laure Gagez , Sophie Sablé , Laurent Picot , Valérie Thiéry , Andrew E. H. Wheatley , Philippe C. Gros , Florence Mongin

Tetrahedron, 2013, 69 (47), pp.10123-10133. ⟨10.1016/j.tet.2013.09.030⟩

Measuring Angiotensin-I Converting Enzyme Inhibitory Activity by Micro Plate Assays: Comparison Using Marine Cryptides and Tentative Threshold Determinations with Captopril and Losartan

Yesmine Ben Henda , Anis Labidi , Ingrid Arnaudin , Nicolas Bridiau , Régis Delatouche , Thierry Maugard , Jean-Marie Piot , Frédéric Sannier , Valérie Thiery , Stéphanie Bordenave-Juchereau

Journal of Agricultural and Food Chemistry, 2013, 61 (45), pp.10685-10690

Cathepsin D activity and selectivity in the acidic conditions of a tumor microenvironment: Utilization in the development of a novel Cathepsin D substrate for simultaneous cancer diagnosis and therapy

Oussama Achour , Nicolas Bridiau , Meriem Kacem , Régis Delatouche , Stéphanie Bordenave-Juchereau , Frédéric Sannier , Valérie Thiery , Jean-Marie Piot , Thierry Maugard , Ingrid Arnaudin

Biochimie, 2013, 95 (11), pp.2010-2017

Antiproliferative Activity of Cyanophora paradoxa Pigments in Melanoma, Breast and Lung Cancer Cells

Paul-Hubert Baudelet , Anne-Laure Gagez , Jean-Baptiste Bérard , Camille Juin , Nicolas Bridiau , Raymond Kaas , Valérie Thiéry , Jean-Paul Cadoret , Laurent Picot

Marine drugs, 2013, 11 (11), pp.4390-4406

Towards the Clinical Use of Phytoplankton Carotenoid Pigments to Cure Cancer

Camille Juin , Valérie Thiéry , Jean-Paul Cadoret , Laurent Picot

oceanography, open access, 2013, 1 (3), ⟨10.4172/2332-2632.1000e105⟩

2012

Article dans une revue

One-Pot Synthesis of Pyrrolo[1,2‑a]quinoxaline Derivatives via Iron-Promoted Aryl Nitro Reduction and Aerobic Oxidation of Alcohols

Maria Pereira , Valérie Thiéry

Organic Letters, 2012, 14, pp.4754-4757. ⟨10.1021/ol302006b⟩

Communication dans un congrès

Aide au ciblage du microenvironnement tumoral par le développement d'un nano-système de détection et de traitement de tumeurs visant l'inhibition spécifique de l'héparanase

Azza Ghodhbani , Meriem Kacem , Oussama Achour , Florian Le Joubioux , Régis Delatouche , Nicolas Bridiau , Valérie Thiéry , Jean-Marie Piot , Thierry Maugard , Ingrid Fruitier-Arnaudin

Journées de la Section Régionale Centre-Ouest de la Société Chimique de France, Dec 2012, Poitiers, France

2011

Article dans une revue

Antiproliferative Activity of Violaxanthin Isolated from Bioguided Fractionation of Dunaliella tertiolecta Extracts

Virginie Pasquet , Perrine Morisset , Saïd Ihammouine , Amandine Chepied , Lucie Aumailley , Jean-Baptiste Bérard , Benoît Serive , Raymond Kaas , Isabelle Lanneluc , Valérie Thiéry , Mathieu Lafferriere , Jean-Marie Piot , Thierry Patrice , Jean-Paul Cadoret , Laurent Picot

Marine drugs, 2011, 9 (5), pp.819-831. ⟨10.3390/md9050819⟩

Antiproliferative Activity of Violaxanthin Isolated from Bioguided Fractionation of Dunaliella tertiolecta Extracts

Virginie Pasquet , Perrine Morisset , Saïd Ihammouine , Amandine Chepied , Lucie Aumailley , Jean-Baptiste Bérard , Benoît Serive , Raymond Kaas , Isabelle Lanneluc , Valérie Thiéry , Mathieu Lafferière , Jean-Marie Piot , Thierry Patrice , Jean-Paul Cadoret , Laurent Picot

Marine drugs, 2011, 9, pp.819-831. ⟨10.3390/md9050819⟩

2009

Article dans une revue

Synthesis and kinase inhibitory activity of novel substituted indigoids

Anne Beauchard , Helene Laborie , Hervé Rouillard , Olivier Lozach , Yoan Ferandin , Rémy Le Guével , Christiane Guguen-Guillouzo , Laurent Meijer , Thierry Besson , Valérie Thiéry

Bioorganic and Medicinal Chemistry Letters, 2009, 17 (17), pp.6257-6263. ⟨10.1016/j.bmc.2009.07.051⟩

Synthesis and kinase inhibitory activity of novel substituted indigoids.

Anne Beauchard , Hélène Laborie , Hervé Rouillard , Olivier Lozach , Yoan Ferandin , Rémy Le Guével , Christiane Guguen-Guillouzo , Laurent Meijer , Thierry Besson , Valérie Thiéry

Bioorganic and Medicinal Chemistry, 2009, 17 (17), pp.6257-63. ⟨10.1016/j.bmc.2009.07.051⟩

2008

Article dans une revue

Synthesis and evaluation of the antimicrobial activity of novel quinazolinones

Maria de Fatima Pereira , Romain Chevrot , Eric Rosenfeld , Valérie Thiéry , Thierry Besson

Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 22 (5), pp.577-583. ⟨10.1080/14756360701425345⟩

Microwave-assisted Synthesis of Novel Thiazolocarbazoles and Evaluation as Potential Anticancer Agents. Part III

Alexandra Testard , Laurent Picot , Ingrid Fruitier-Arnaudin , Jean-Marie Piot , Hadjila Chabane , Lisianne Domon , Valérie Thiery , Thierry Besson

Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 19 (6), pp.467-473. ⟨10.1080/14756360412331280491⟩

Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies

Cédric Logé , Alexandra Testard , Valérie Thiéry , Olivier Lozach , Mélina Blairvacq , Jean-Michel Robert , Laurent Meijer , Thierry Besson

European Journal of Medicinal Chemistry, 2008, 43 (7), pp.1469-1477. ⟨10.1016/j.ejmech.2007.09.020⟩

2006

Article dans une revue

Synthesis of novel 5-substituted indirubins as protein kinases inhibitors

Anne Beauchard , Yoan Ferandin , Stéphane Frère , Olivier Lozach , Mélina Blairvacq , Laurent Meijer , Valérie Thiéry , Thierry Besson

Bioorganic and Medicinal Chemistry, 2006, 14 (18), pp.6434-43. ⟨10.1016/j.bmc.2006.05.036⟩

Thiazolo[5,4-f]quinazolin-9-ones, inhibitors of glycogen synthase kinase-3

Alexandra Testard , Cédric Logé , Benoît Léger , Jean-Michel Robert , Olivier Lozach , Mélina Blairvacq , Laurent Meijer , Valérie Thiéry , Thierry Besson

Bioorganic and Medicinal Chemistry Letters, 2006, 16 (13), pp.3419-3423. ⟨10.1016/j.bmcl.2006.04.006⟩

Synthesis of novel 2,3-condensed thieno[2,3- d ]pyrimidin-4-ones via Appel's salt chemistry

Maria de Fatima Pereira , Valérie Thiéry , Thierry Besson

Journal of Sulfur Chemistry, 2006, 27 (1), pp.49-55. ⟨10.1080/17415990500493213⟩

2005

Article dans une revue

Synthesis and evaluation of the antiproliferative activity of novel thiazoloquinazolinone kinases inhibitors.

Alexandra Testard , Laurent Picot , Olivier Lozach , Melina Blairvacq , Laurent Meijer , Laurence Murillo , Jean-Marie Piot , Valérie Thiéry , Thierry Besson

Journal of Enzyme Inhibition and Medicinal Chemistry, 2005, 20 (6), pp.557-568. ⟨10.1080/14756360500212399⟩

2003

Article dans une revue

Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles

Stéphane Frère , Valérie Thiéry , Thierry Besson

Synthetic Communications, 2003, 33 (21), pp.3795-3804. ⟨10.1081/SCC-120025190⟩

Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles

Valérie Thiéry , Thierry Besson

Synthetic Communications, 2003, 33 (21), pp.3795-3804. ⟨10.1081/SCC-120025190⟩

2002

Article dans une revue

Efficient solvent-free microwave phosphorylation of microcrystalline cellulose

Natalia Gospodinova , Axelle Grelard , Marc Jeannin , Gabrielle Chitanu , Adrian Carpov , Valérie Thiéry , Thierry Besson

Green Chemistry, 2002, 4 (3), pp.220-222. ⟨10.1039/b200295g⟩

2000

Article dans une revue

Imidazoquinolinethiones from 8-aminoquinolines by a novel peri-participation

Thierry Besson , Charles Rees , David Roe , Valérie Thiéry

Journal of the Chemical Society, Perkin Transactions 1, 2000, 4, pp.555-561. ⟨10.1039/a908952g⟩

1998

Article dans une revue

N-(Cyanothioformyl)indoline; a new indoline ring forming reaction

Thierry Besson , Gerald Guillaumet , Christelle Lamazzi , Charles Rees , Valérie Thiéry

Journal of the Chemical Society, Perkin Transactions 1, 1998