Thiéry Valérie

Enseignant-chercheur, Professeur
Université de La Rochelle
Section de Recherche : CNU 32
Institut scientifique du CNRS référent : INEE

Mots clés : Hétérocycles, alcaloïde, chimie verte, micro-onde

  • Responsable du groupe de chimie organique
  • Correspondant Hygiène et Sécurité de LIENSs-CURIE
Thèmes de Recherche.
  • Chimie hétérocyclique (N,O,S), étude de la réactivité des iminodithiazoles
  • Synthèse d’analogues d’alcaloïdes marins à visée antitumorales
  • Synthèse d’inhibiteurs de kinases
  • Chimie assistée- par micro-ondes : nouvelles méthodologies de synthèse, extraction
  • Synthèse asymétrique

Liste des publications :

60 résultats

2024

Article dans une revue

Contribution of Professor Charles Rees to the development of the chemistry of disulfur dichloride
Thierry Besson , Lidia S Konstntinova , Panayiotis A Koutentis , Oleg A Rakitin , Sivaprasad Sivadasan , Valérie Thiéry , Tomás Torroba
ARKIVOC - Online Journal of Organic Chemistry, 2024, Commemorative Issue in Honor of Prof. Alan R. Katritzky and Prof. Charles Rees on the occasion of the 25th anniversary of the first publication of Arkivoc (Archive for Organic Chemistry), 2024 (1), ⟨10.24820/ark.5550190.p012.136⟩
Contribution of Professor Charles W. Rees to the development of the chemistry of disulfur dichloride
Thierry Besson , Lidia Konstantinova , Panayiotis Koutentis , Oleg Rakitin , Sivaprasad Sivadasan , Valérie Thiéry , Tomás Torroba
ARKIVOC - Online Journal of Organic Chemistry, 2024, 2024 (1), ⟨10.24820/ark.5550190.p012.136⟩
Deprotonative Metallation of Benzofuran and Benzothiophene Derivatives for the Formation of Tetracyclic and Pentacyclic Heteroaromatic Compounds
Loubna Elmir , Ghenia Bentabed-Ababsa , William Erb , Thierry Roisnel , Jean-Pierre Hurvois , Laurent Picot , Valérie Thiéry , Florence Mongin
European Journal of Organic Chemistry, In press, ⟨10.1002/ejoc.202400374⟩

2023

Article dans une revue

From benzofuro-, benzothieno- and 10-methylindolo-[2,3-b]-fused benzothiopyrano[4,3,2-de]quinolines to the corresponding benzothiopyrano[4,3,2-de]1,8-naphthyridines: synthesis and properties of these hexacyclic heteroaromatic compounds
Nicolas Mast , William Erb , Lionel Nauton , Pascale Moreau , Olivier Mongin , Thierry Roisnel , Margaux Macaigne , Thomas Robert , Stéphane Bach , Laurent Picot , Valérie Thiéry , Jean-Pierre Hurvois , Florence Mongin
New Journal of Chemistry, 2023, 47 (1), pp.258-283. ⟨10.1039/D2NJ04567B⟩
A review of phototoxic plants, their phototoxic metabolites, and possible developments as photosensitizers.
Raphaelle Petit , Jonathan Izambart , Mathieu Guillou , Jackson Guedes da Silva Almeida , Raimundo Gonçalves de Oliveira Junior , Vincent Sol , Tan-Sothea Ouk , Raphael Grougnet , Lucindo Quintans-Junior , Przemyslaw Sitarek , Valérie Thiéry , Laurent Picot
Chemistry and Biodiversity, 2023, ⟨10.1002/cbdv.202300494⟩

2022

Article dans une revue

Bisphosphonylallenes as Suitable Scaffolds for Unprecedented 4,5-Diphosphonyldihydropyridazines and 3,4-Diphosphonylpyrroles Displaying Antimelanoma Activity
Kmar Abaid , William Erb , David Virieux , Laurent Picot , Benjamin Musnier , Valérie Thiéry , Thierry Roisnel , Florence Mongin , Soufiane Touil
ACS Omega, 2022, 7 (43), pp.38894-38901. ⟨10.1021/acsomega.2c04619⟩
Archaea Carotenoids: Natural Pigments with Unexplored Innovative Potential
Antoine Grivard , Isabelle Goubet , Luiz Miranda de Souza Duarte Filho , Valérie Thiéry , Sylvie Chevalier , Raimundo Gonçalves de Oliveira Júnior , Noureddine El Aouad , Jackson Roberto Guedes da Silva Almeida , Przemysław Sitarek , Lucindo José Quintans-Junior , Raphaël Grougnet , Hélène Agogué , Laurent Picot
Marine drugs, 2022, Marine Pigments, 20 (8), pp.524. ⟨10.3390/md20080524⟩
Alterins, a new family of marine antibacterial cyclolipopeptides
Clément Offret , Héléna Cuny , Pierre-Edouard Bodet , Florie Desriac , Camille Jegou , Alexis Bazire , Romain Chevrot , Valérie Thiery , Benjamin Brillet , Yannick Fleury
International Journal of Antimicrobial Agents, 2022, pp.106514. ⟨10.1016/j.ijantimicag.2021.106514⟩

2021

Article dans une revue

Thiazolo[5,4- f ]quinoxalines, Oxazolo[5,4- f ]quinoxalines and Pyrazino[ b,e ]isatins: Synthesis from 6-Aminoquinoxalines and Properties
Frédéric Lassagne , Joshua M. Sims , William Erb , Olivier Mongin , Nicolas Richy , Nour El Osmani , Ziad Fajloun , Laurent Picot , Valérie Thiéry , Thomas Robert , Stéphane Bach , Vincent Dorcet , Thierry Roisnel , Florence Mongin
European Journal of Organic Chemistry, 2021, 2021 (19), pp.2756-2763. ⟨10.1002/ejoc.202100362⟩
The Franco-Brazilian network on natural products (FB2NP): a new network promoting cooperation and exchanges in natural products research
Jackson Almeida , Raphaël Grougnet , Lucindo Quintans , Sylvie Chevalier , Marc Feuilloley , Thomas Robert , Stéphane Bach , Raimundo Oliveira , Valérie Thiéry , Jean-Pierre Bazureau , Florence Mongin , Marina Kritsanida , Vincent Sol , Vicente Costa , Nathalie Bourgougnon , Pascal Marchand , Laurent Picot
Iodothiophenes and Related Compounds as Coupling Partners in Copper-Mediated N-Arylation of Anilines
Salima Bouarfa , Ghenia Bentabed-Ababsa , William Erb , Laurent Picot , Valérie Thiéry , Thierry Roisnel , Vincent Dorcet , Florence Mongin
Synthesis: Journal of Synthetic Organic Chemistry, 2021, 53 (07), pp.1271-1284. ⟨10.1055/s-0040-1706542⟩

2020

Article dans une revue

2-Aminobenzaldehyde, a common precursor to acridines and acridones endowed with bioactivities
Sarah Zeghada , Ghenia Bentabed-Ababsa , Olivier Mongin , William Erb , Laurent Picot , Valérie Thiéry , Thierry Roisnel , Vincent Dorcet , Florence Mongin
Tetrahedron, 2020, 76 (38), pp.131435. ⟨10.1016/j.tet.2020.131435⟩
Carotenoids from Rhodomonas salina Induce Apoptosis and Sensitize A2058 Melanoma Cells to Chemotherapy
Raimundo Gonçalves de Oliveira-Júnior , Elodie Nicolau , Antoine Bonnet , Grégoire Prunier , Laureen Beaugeard , Nicolas Joguet , Valérie Thiéry , Laurent Picot
Revista Brasileira de Farmacognosia, 2020, 30 (2), pp.155-168. ⟨10.1007/s43450-020-00036-2⟩
Functionalization of 9-thioxanthone at the 1-position: From arylamino derivatives to [1]benzo(thio)pyrano[4,3,2-de]benzothieno[2,3-b]quinolines of biological interest
Nahida Mokhtari Brikci-Nigassa , Lionel Nauton , Pascale Moreau , Olivier Mongin , Raphael E Duval , Laurent Picot , Valérie Thiery , Mohamed Souab , Blandine Baratte , Sandrine Ruchaud , Stéphane Bach , Rémy Le Guével , Ghenia Bentabed-Ababsa , William Erb , Thierry Roisnel , Vincent Dorcet , Florence Mongin
Bioorganic Chemistry, 2020, 94, pp.103347. ⟨10.1016/j.bioorg.2019.103347⟩

2019

Article dans une revue

Characterisation of the anti-migratory activity of the 6-bromoindirubin-3’oxime (BIO) derivative VTIND42 in patient-derived GBM subpopulations
Samuel Peat , Anke Bruning-Richardson , Laurent Meijer , Sean Lawler , Valérie Thiéry , Ruth Morton
Neuro-Oncology, 2019, 21 (Supplement_4), pp.iv6-iv7. ⟨10.1093/neuonc/noz167.026⟩
Crystal Structure of 6,7-Dihydro-5a,7a,13,14-tetraaza-pentaphene-5,8-dione
Jean Guillon , Maria de Fatima Pereira-Rosenfeld , Noël Pinaud , Thierry Besson , Valérie Thiéry , Laurent Picot , Mathieu Marchivie
X-Ray Structure Analysis Online, 2019, 35 (10), pp.57-59. ⟨10.2116/xraystruct.35.57⟩

2018

Article dans une revue

Complete Genome Sequence of the Polymyxin E (Colistin)-Producing Paenibacillus sp. Strain B-LR
Caroline Salsano , Sandrine Didelot , Fatoumata Tambadou , Thibault Caradec , Valérie Sopena , Cyrille Barthélémy , Valérie Thiéry , Romain Chevrot
Microbiology Resource Announcements, 2018, 7 (23), ⟨10.1128/MRA.01013-18⟩
From Quinoxaline, Pyrido[2,3-b]pyrazine and Pyrido[3,4-b]pyrazine to Pyrazino-Fused Carbazoles and Carbolines
Frédéric Lassagne , Timothy Langlais , Elsa Caytan , Emmanuelle Limanton , Ludovic Paquin , Manon Boullard , Coline Courtel , Idriss Curbet , Clément Gédéon , Julien Lebreton , Laurent Picot , Valérie Thiéry , Mohamed Souab , Blandine Baratte , Sandrine Ruchaud , Stéphane Bach , Thierry Roisnel , Florence Mongin
Molecules, 2018, 23 (11), pp.2961. ⟨10.3390/molecules23112961⟩
Sensitization of tumor cells to chemotherapy by natural products: a systematic review of preclinical data and molecular mechanisms
Raimundo Gonçalves de Oliveira Júnior , Christiane Adrielly Alves Ferraz , Jackson Roberto Guedes da Silva Almeida , Raphäel Grougnet , Valérie Thiéry , Laurent Picot
Fitoterapia, 2018, 129, pp.383-400. ⟨10.1016/j.fitote.2018.02.025⟩
Synthesis of 2-Mercapto-(2-Oxoindolin-3-Ylidene)Acetonitriles from 3-(4-Chloro-5H-1,2,3-Dithiazol-5-Ylidene)Indolin-2-ones
Boris Letribot , Régis Delatouche , Hervé Rouillard , Antoine Bonnet , Jean-René Chérouvrier , Lisianne Domon , Thierry Besson , Valérie Thiéry
Molecules, 2018, 23 (6), pp.1390. ⟨10.3390/molecules23061390⟩
2-Aminophenones, a common precursor to N-aryl isatins and acridines endowed with bioactivities
Nahida Mokhtari Brikci-Nigassa , Ghenia Bentabed-Ababsa , William Erb , Floris Chevallier , Laurent Picot , Lucille Vitek , Audrey Fleury , Valérie Thiéry , Mohamed Souab , Thomas Robert , Sandrine Ruchaud , Stéphane Bach , Thierry Roisnel , Florence Mongin
Tetrahedron, 2018, 74 (15), pp.1785-1801. ⟨10.1016/j.tet.2018.02.038⟩
Zeaxanthin from Porphyridium purpureum induces apoptosis in human melanoma cells expressing the oncogenic BRAF V600E mutation and sensitizes them to the BRAF inhibitor vemurafenib
Camille Juin , Raimundo Gonçalves de Oliveira Junior , Audrey Fleury , Chloé Oudinet , Lior Pytowski , Jean-Baptiste Bérard , Elodie Nicolau , Valérie Thiéry , Isabelle Lanneluc , Laureen Beaugeard , Grégoire Prunier , Jackson Roberto Guedes da Silva Almeida , Laurent Picot
Revista Brasileira de Farmacognosia, 2018, 28 (4), pp.457-467. ⟨10.1016/j.bjp.2018.05.009⟩

2017

Article dans une revue

Synthesis of novel heterocyclic fused pyrimidin-4-one derivatives from imino-1,2,3-dithiazoles
Maria de Fatima Pereira , Elena Sarghe , Hervé Rouillard , Lisianne Domon , Jean-René Chérouvrier , Valérie Thiéry , Jacques Royer
ARKIVOC - Online Journal of Organic Chemistry, 2017, 2017 (3), pp.335-345. ⟨10.24820/ark.5550190.p010.256⟩
Antimelanoma activity of Heterocapsa triquetra pigments
Quentin Haguet , Antoine Bonnet , Jean-Baptiste Bérard , Joelle Goldberg , Nicolas Joguet , Audrey Fleury , Valérie Thiéry , Laurent Picot
Algal Research - Biomass, Biofuels and Bioproducts, 2017, 25, pp.207 - 215. ⟨10.1016/j.algal.2017.04.034⟩

2016

Article dans une revue

Improved racemate resolution of pentan-2-ol and trans-(Z)-cyclooct-5-ene-1,2-diol by lipase catalysis
Marianne Graber , Hervé Rouillard , Régis Delatouche , Najla Fniter , Belsem Belkhiria , Antoine Bonnet , Lisiane Domon , Valérie Thiéry
Journal of Biotechnology, 2016, 238, pp.60-68. ⟨10.1016/j.jbiotec.2016.09.010⟩
Could Fucoxanthin Interaction with Lipid Rafts Mediate its Cytotoxicity in Cancer Cells?
Raimundo Gonçalves Oliveira-Junior , Valérie Thiéry , Odile Sergent , Martine Chevanne , Laurent Picot
Journal of Oceanography and Marine Research, 2016, 4 (1), pp.1000144. ⟨10.4172/jomr.1000144⟩

2015

Article dans une revue

Azine and Diazine Functionalization Using 2,2,6,6-Tetramethylpiperidino-Based Lithium–Metal Combinations: Application to the Synthesis of 5,9-Disubstituted Pyrido[3′,2′:4,5]pyrrolo[1,2-c] pyrimidines
Nada Marquise , Tan Tai Nguyen , Floris Chevallier , Laurent Picot , Valérie Thiéry , Olivier Lozach , Stéphane Bach , Sandrine Ruchaud , Florence Mongin
SYNLETT, 2015, 26 (20), pp.2811-2816. ⟨10.1055/s-0035-1560496⟩
Deproto-metallation of N-arylated pyrroles and indoles using a mixed lithium–zinc base and regioselectivity-computed CH acidity relationship
Mohamed Yacine Ameur Messaoud , Ghenia Bentabed-Ababsa , Madani Hedidi , Aïcha Derdour , Floris Chevallier , Yury S. Halauko , Oleg A. Ivashkevich , Vadim E. Matulis , Laurent Picot , Valérie Thiéry , Thierry Roisnel , Vincent Dorcet , Florence Mongin
Beilstein Journal of Organic Chemistry, 2015, 11, pp.1475-1485. ⟨10.3762/bjoc.11.160⟩
Caractérisations analytiques des extraits colorants des plantes tinctoriales d'Afrique Centrale
A.B. Madiélé , Jean-Michel Zhao , Valérie Thiéry , Huguette Agnaniet , Christine Brunet , Marianne Graber , Jean-Maurille Ouamba
Lebanese Science Journal, 2015, 16, pp.33-44
Characterization of the colistin (polymyxin E1 and E2) biosynthetic gene cluster.
Fatoumata Tambadou , Thibault Caradec , Anne-Laure Gagez , Antoine Bonnet , Valérie Sopena , Nicolas Bridiau , Valérie Thiéry , Sandrine Didelot, , Cyrille Barthélémy , Romain Chevrot
Archives of Microbiology, 2015, 197 (4), pp.521-532. ⟨10.1007/s00203-015-1084-5⟩
Microwave-Assisted Extraction of Phycobiliproteins from Porphyridium purpureum.
Camille Juin , Jean-René Chérouvrier , Valérie Thiery , Anne-Laure Gagez , Jean-Baptiste Bérard , Nicolas, Joguet , Raymond Kaas , Jean-Paul Cadoret , Laurent Picot
Biotechnology and Applied Biochemistry, 2015, ⟨10.1007/s12010-014-1250-2⟩
UPLC-MSE Profiling of Phytoplankton Metabolites: Application to the Identification of Pigments and Structural Analysis of Metabolites in Porphyridium purpureum
Camille Juin , Antoine Bonnet , Elodie Nicolau , Jean-Baptiste Bérard , Devillers, Romain , Valérie Thiéry , Jean-Paul Cadoret , Laurent Picot
Marine drugs, 2015, 13 (4), pp.1541-2558. ⟨10.3390/md13042541⟩

2014

Article dans une revue

Microwave-Assisted Kinetic Resolution of Homochiral (Z)-Cyclooct-5-ene-1,2-diol and (Z)-2-Acetoxycyclooct-4-enyl Acetate Using Lipases
Hervé Rouillard , Emmanuel Deau , Lisiane Domon , Jean-René Chérouvrier , Marianne Graber , Valérie Thiéry
Molecules, 2014, 19, pp.9215-9227. ⟨10.3390/molecules19079215⟩
Novel nonribosomal peptide synthetase (NRPS) genes sequenced from intertidal mudflat bacteria
Fatoumata Tambadou , Isabelle Lanneluc , Sophie Sablé , Géraldine Klein , Ibtissem Doghri , Valérie Sopena , Sandrine Didelot , Cyrille Barthélémy , Valérie Thiéry , Romain Chevrot
FEMS Microbiology Letters, 2014, pp.n/a-n/a. ⟨10.1111/1574-6968.12532⟩
Synthesis of C,N'-linked bis-heterocycles using a deprotometalation-iodination-N-arylation sequence and evaluation of their antiproliferative activity in melanoma cells
Madani Hedidi , Ghenia Bentabed-Ababsa , Aicha Derdour , Thierry Roisnel , Vincent Dorcet , Floris Chevallier , Laurent Picot , Valérie Thiery , Mongin Florence
Bioorganic and Medicinal Chemistry, 2014, 22 (13), pp.3498-3507. ⟨10.1016/j.bmc.2014.04.028⟩

2013

Article dans une revue

Synthesis of azafluorenones and related compounds using deprotocupration-aroylation followed by intramolecular direct arylation
Nada Marquise , Philip J. Harford , Floris Chevallier , Thierry Roisnel , Vincent Dorcet , Anne-Laure Gagez , Sophie Sablé , Laurent Picot , Valérie Thiéry , Andrew E. H. Wheatley , Philippe C. Gros , Florence Mongin
Tetrahedron, 2013, 69 (47), pp.10123-10133. ⟨10.1016/j.tet.2013.09.030⟩
Measuring Angiotensin-I Converting Enzyme Inhibitory Activity by Micro Plate Assays: Comparison Using Marine Cryptides and Tentative Threshold Determinations with Captopril and Losartan
Yesmine Ben Henda , Anis Labidi , Ingrid Arnaudin , Nicolas Bridiau , Régis Delatouche , Thierry Maugard , Jean-Marie Piot , Frédéric Sannier , Valérie Thiery , Stéphanie Bordenave-Juchereau
Journal of Agricultural and Food Chemistry, 2013, 61 (45), pp.10685-10690
Antiproliferative Activity of Cyanophora paradoxa Pigments in Melanoma, Breast and Lung Cancer Cells
Paul-Hubert Baudelet , Anne-Laure Gagez , Jean-Baptiste Berard , Camille Juin , Nicolas Bridiau , Raymond Kaas , Valerie Thiery , Jean-Paul Cadoret , Laurent Picot
Marine drugs, 2013, 11 (11), pp.4390-4406. ⟨10.3390/md11114390⟩
Cathepsin D activity and selectivity in the acidic conditions of a tumor microenvironment: Utilization in the development of a novel Cathepsin D substrate for simultaneous cancer diagnosis and therapy
Oussama Achour , Nicolas Bridiau , Meriem Kacem , Régis Delatouche , Stéphanie Bordenave-Juchereau , Frédéric Sannier , Valérie Thiery , Jean-Marie Piot , Thierry Maugard , Ingrid Arnaudin
Biochimie, 2013, 95 (11), pp.2010-2017
Antiproliferative Activity of Cyanophora paradoxa Pigments in Melanoma, Breast and Lung Cancer Cells
Paul-Hubert Baudelet , Anne-Laure Gagez , Jean-Baptiste Bérard , Camille Juin , Nicolas Bridiau , Raymond Kaas , Valérie Thiéry , Jean-Paul Cadoret , Laurent Picot
Marine drugs, 2013, 11 (11), pp.4390-4406
Towards the Clinical Use of Phytoplankton Carotenoid Pigments to Cure Cancer
Camille Juin , Valérie Thiéry , Jean-Paul Cadoret , Laurent Picot
oceanography, open access, 2013, 1 (3), ⟨10.4172/2332-2632.1000e105⟩

2012

Article dans une revue

One-Pot Synthesis of Pyrrolo[1,2‑a]quinoxaline Derivatives via Iron-Promoted Aryl Nitro Reduction and Aerobic Oxidation of Alcohols
Maria Pereira , Valérie Thiéry
Organic Letters, 2012, 14, pp.4754-4757. ⟨10.1021/ol302006b⟩

Communication dans un congrès

Aide au ciblage du microenvironnement tumoral par le développement d'un nano-système de détection et de traitement de tumeurs visant l'inhibition spécifique de l'héparanase
Azza Ghodhbani , Meriem Kacem , Oussama Achour , Florian Le Joubioux , Régis Delatouche , Nicolas Bridiau , Valérie Thiéry , Jean-Marie Piot , Thierry Maugard , Ingrid Fruitier-Arnaudin
Journées de la Section Régionale Centre-Ouest de la Société Chimique de France, Dec 2012, Poitiers, France

2011

Article dans une revue

Antiproliferative Activity of Violaxanthin Isolated from Bioguided Fractionation of Dunaliella tertiolecta Extracts
Virginie Pasquet , Perrine Morisset , Saïd Ihammouine , Amandine Chepied , Lucie Aumailley , Jean-Baptiste Bérard , Benoît Serive , Raymond Kaas , Isabelle Lanneluc , Valérie Thiéry , Mathieu Lafferriere , Jean-Marie Piot , Thierry Patrice , Jean-Paul Cadoret , Laurent Picot
Marine drugs, 2011, 9 (5), pp.819-831. ⟨10.3390/md9050819⟩
Antiproliferative Activity of Violaxanthin Isolated from Bioguided Fractionation of Dunaliella tertiolecta Extracts
Virginie Pasquet , Perrine Morisset , Saïd Ihammouine , Amandine Chepied , Lucie Aumailley , Jean-Baptiste Bérard , Benoît Serive , Raymond Kaas , Isabelle Lanneluc , Valérie Thiéry , Mathieu Lafferière , Jean-Marie Piot , Thierry Patrice , Jean-Paul Cadoret , Laurent Picot
Marine drugs, 2011, 9, pp.819-831. ⟨10.3390/md9050819⟩
Study on the microalgal pigments extraction process: Performance of microwave assisted extraction
Virginie Pasquet , Jean-Rene Cherouvrier , Firas Farhat , Valerie Thiery , Jean-Marie Piot , Jean-Baptiste Berard , Raymond Kaas , Benoit Serive , Thierry Patrice , Jean-Paul Cadoret , Laurent Picot
Process Biochemistry, 2011, 46 (1), pp.59-67. ⟨10.1016/j.procbio.2010.07.009⟩

2009

Article dans une revue

Synthesis and kinase inhibitory activity of novel substituted indigoids.
Anne Beauchard , Hélène Laborie , Hervé Rouillard , Olivier Lozach , Yoan Ferandin , Rémy Le Guével , Christiane Guguen-Guillouzo , Laurent Meijer , Thierry Besson , Valérie Thiéry
Bioorganic and Medicinal Chemistry, 2009, 17 (17), pp.6257-63. ⟨10.1016/j.bmc.2009.07.051⟩
Synthesis and kinase inhibitory activity of novel substituted indigoids
Anne Beauchard , Helene Laborie , Hervé Rouillard , Olivier Lozach , Yoan Ferandin , Rémy Le Guével , Christiane Guguen-Guillouzo , Laurent Meijer , Thierry Besson , Valérie Thiéry
Bioorganic and Medicinal Chemistry Letters, 2009, 17 (17), pp.6257-6263. ⟨10.1016/j.bmc.2009.07.051⟩

2008

Article dans une revue

Synthesis and evaluation of the antimicrobial activity of novel quinazolinones
Maria de Fatima Pereira , Romain Chevrot , Eric Rosenfeld , Valérie Thiéry , Thierry Besson
Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 22 (5), pp.577-583. ⟨10.1080/14756360701425345⟩
Microwave-assisted Synthesis of Novel Thiazolocarbazoles and Evaluation as Potential Anticancer Agents. Part III
Alexandra Testard , Laurent Picot , Ingrid Fruitier-Arnaudin , Jean-Marie Piot , Hadjila Chabane , Lisianne Domon , Valérie Thiery , Thierry Besson
Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 19 (6), pp.467-473. ⟨10.1080/14756360412331280491⟩
Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1)/glycogen synthase kinase-3 (GSK-3) inhibitors: Synthesis, biological evaluation and molecular modeling studies
Cédric Logé , Alexandra Testard , Valérie Thiéry , Olivier Lozach , Mélina Blairvacq , Jean-Michel Robert , Laurent Meijer , Thierry Besson
European Journal of Medicinal Chemistry, 2008, 43 (7), pp.1469-1477. ⟨10.1016/j.ejmech.2007.09.020⟩

2006

Article dans une revue

Synthesis of novel 5-substituted indirubins as protein kinases inhibitors
Anne Beauchard , Yoan Ferandin , Stéphane Frère , Olivier Lozach , Mélina Blairvacq , Laurent Meijer , Valérie Thiéry , Thierry Besson
Bioorganic and Medicinal Chemistry, 2006, 14 (18), pp.6434-43. ⟨10.1016/j.bmc.2006.05.036⟩
Thiazolo[5,4-f]quinazolin-9-ones, inhibitors of glycogen synthase kinase-3
Alexandra Testard , Cédric Logé , Benoît Léger , Jean-Michel Robert , Olivier Lozach , Mélina Blairvacq , Laurent Meijer , Valérie Thiéry , Thierry Besson
Bioorganic and Medicinal Chemistry Letters, 2006, 16 (13), pp.3419-3423. ⟨10.1016/j.bmcl.2006.04.006⟩
Synthesis of novel 2,3-condensed thieno[2,3- d ]pyrimidin-4-ones via Appel's salt chemistry
Maria de Fatima Pereira , Valérie Thiéry , Thierry Besson
Journal of Sulfur Chemistry, 2006, 27 (1), pp.49-55. ⟨10.1080/17415990500493213⟩

2005

Article dans une revue

Synthesis and evaluation of the antiproliferative activity of novel thiazoloquinazolinone kinases inhibitors.
Alexandra Testard , Laurent Picot , Olivier Lozach , Melina Blairvacq , Laurent Meijer , Laurence Murillo , Jean-Marie Piot , Valérie Thiéry , Thierry Besson
Journal of Enzyme Inhibition and Medicinal Chemistry, 2005, 20 (6), pp.557-568. ⟨10.1080/14756360500212399⟩

2003

Article dans une revue

Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles
Stéphane Frère , Valérie Thiéry , Thierry Besson
Synthetic Communications, 2003, 33 (21), pp.3795-3804. ⟨10.1081/SCC-120025190⟩
Eco-Friendly Microwave-Assisted Scaleable Synthesis of 2-Cyanobenzothiazoles via N -Arylimino-1,2,3-dithiazoles
Valérie Thiéry , Thierry Besson
Synthetic Communications, 2003, 33 (21), pp.3795-3804. ⟨10.1081/SCC-120025190⟩

2002

Article dans une revue

Efficient solvent-free microwave phosphorylation of microcrystalline cellulose
Natalia Gospodinova , Axelle Grelard , Marc Jeannin , Gabrielle Chitanu , Adrian Carpov , Valérie Thiéry , Thierry Besson
Green Chemistry, 2002, 4 (3), pp.220-222. ⟨10.1039/b200295g⟩

2000

Article dans une revue

Imidazoquinolinethiones from 8-aminoquinolines by a novel peri-participation
Thierry Besson , Charles Rees , David Roe , Valérie Thiéry
Journal of the Chemical Society, Perkin Transactions 1, 2000, 4, pp.555-561. ⟨10.1039/a908952g⟩

1998

Article dans une revue

N-(Cyanothioformyl)indoline; a new indoline ring forming reaction
Thierry Besson , Gerald Guillaumet , Christelle Lamazzi , Charles Rees , Valérie Thiéry
Journal of the Chemical Society, Perkin Transactions 1, 1998